Research output per year
Research output per year
- 13 results
Search results
-
2023
Enolase Inhibitors as Early Lead Therapeutics against Trypanosoma brucei
Roster, C. P., LaVigne, D., Milanes, J. E., Knight, E., Anderson, H. D., Pizarro, S., Harding, E. M., Morris, M. T., Yan, V. C., Pham, C. D., Muller, F., Kwain, S., Rees, K. C., Dominy, B., Whitehead, D. C., Uddin, M. N., Millward, S. W. & Morris, J. C., Nov 2023, In: Pathogens. 12, 11, 1290.Research output: Contribution to journal › Article › peer-review
Open Access -
Overexpression of ameloblastin in secretory ameloblasts results in demarcated, hypomineralized opacities in enamel
Chun, Y. H. P., Tan, C., Villanueva, O., Colley, M. E., Quintanilla, T. J., Basiouny, M. S., Hartel, C. A., Critchfield, C. S., Bach, S. B. H., Fajardo, R. J. & Pham, C. D., 2023, In: Frontiers in Physiology. 14, 1233391.Research output: Contribution to journal › Article › peer-review
Open Access -
2022
An Optimized Bioassay for Screening Combined Anticoronaviral Compounds for Efficacy against Feline Infectious Peritonitis Virus with Pharmacokinetic Analyses of GS-441524, Remdesivir, and Molnupiravir in Cats
Cook, S., Wittenburg, L., Yan, V. C., Theil, J. H., Castillo, D., Reagan, K. L., Williams, S., Pham, C. D., Li, C., Muller, F. L. & Murphy, B. G., Nov 2022, In: Viruses. 14, 11, 2429.Research output: Contribution to journal › Article › peer-review
Open Access12 Scopus citations -
Prodrugs of a 1-Hydroxy-2-oxopiperidin-3-yl Phosphonate Enolase Inhibitor for the Treatment of ENO1-Deleted Cancers
Yan, V. C., Pham, C. D., Ballato, E. S., Yang, K. L., Arthur, K., Khadka, S., Barekatain, Y., Shrestha, P., Tran, T., Poral, A. H., Washington, M., Raghavan, S., Czako, B., Pisaneschi, F., Lin, Y. H., Satani, N., Hammoudi, N., Ackroyd, J. J., Georgiou, D. K., Millward, S. W., & 1 others, Oct 27 2022, In: Journal of Medicinal Chemistry. 65, 20, p. 13813-13832 20 p.Research output: Contribution to journal › Article › peer-review
Open Access3 Scopus citations -
Quantification of Phosphonate Drugs by 1H-31P HSQC Shows That Rats Are Better Models of Primate Drug Exposure than Mice
Barekatain, Y., Khadka, S., Harris, K., Delacerda, J., Yan, V. C., Chen, K. C., Pham, C. D., Uddin, M. N., Avritcher, R., Eisenberg, E. J., Kalluri, R., Millward, S. W. & Muller, F. L., Jul 19 2022, In: Analytical Chemistry. 94, 28, p. 10045-10053 9 p.Research output: Contribution to journal › Article › peer-review
4 Scopus citations -
2021
Bioactive secondary metabolites from the mangrove endophytic fungi Nigrospora oryzae
Ola, A. R. B., Lapailaka, T., Wogo, H. E., Henuk, J. B. D., Simamora, A., Mukkun, L., Proksch, P. & Pham, C. D., Apr 1 2021, In: Indonesian Journal of Chemistry. 21, 4, p. 1016-1022 7 p.Research output: Contribution to journal › Article › peer-review
Open Access7 Scopus citations -
2020
Aliphatic amines are viable pro-drug moieties in phosphonoamidate drugs
Yan, V. C., Pham, C. D., Arthur, K., Yang, K. L. & Muller, F. L., Dec 15 2020, In: Bioorganic and Medicinal Chemistry Letters. 30, 24, 127656.Research output: Contribution to journal › Article › peer-review
3 Scopus citations -
An enolase inhibitor for the targeted treatment of ENO1-deleted cancers
Lin, Y. H., Satani, N., Hammoudi, N., Yan, V. C., Barekatain, Y., Khadka, S., Ackroyd, J. J., Georgiou, D. K., Pham, C. D., Arthur, K., Maxwell, D., Peng, Z., Leonard, P. G., Czako, B., Pisaneschi, F., Mandal, P., Sun, Y., Zielinski, R., Pando, S. C., Wang, X., & 11 others, Dec 2020, In: Nature Metabolism. 2, 12, p. 1413-1426 14 p.Research output: Contribution to journal › Article › peer-review
Open Access37 Scopus citations -
Bioreducible Phosphonoamidate Pro-drug Inhibitor of Enolase: Proof of Concept Study
Yan, V. C., Yang, K. L., Ballato, E. S., Khadka, S., Shrestha, P., Arthur, K., Georgiou, D. K., Washington, M., Tran, T., Poral, A. H., Pham, C. D., Yan, M. J. & Muller, F. L., Jul 9 2020, In: ACS Medicinal Chemistry Letters. 11, 7, p. 1484-1489 6 p.Research output: Contribution to journal › Article › peer-review
2 Scopus citations -
2019
Epigenetic modification, co-culture and genomic methods for natural product discovery
Akone, S. H., Pham, C. D., Chen, H., Ola, A. R. B., Ntie-Kang, F. & Proksch, P., Apr 1 2019, In: Physical Sciences Reviews. 4, 4, 20180118.Research output: Contribution to journal › Article › peer-review
13 Scopus citations -
2014
Callyspongiolide, a cytotoxic macrolide from the marine sponge callyspongia sp.
Pham, C. D., Hartmann, R., Böhler, P., Stork, B., Wesselborg, S., Lin, W., Lai, D. & Proksch, P., Jan 3 2014, In: Organic Letters. 16, 1, p. 266-269 4 p.Research output: Contribution to journal › Article › peer-review
Open Access48 Scopus citations -
2013
Aaptamine derivatives from the indonesian sponge Aaptos suberitoides
Pham, C. D., Hartmann, R., Müller, W. E. G., De Voogd, N., Lai, D. & Proksch, P., Jan 25 2013, In: Journal of Natural Products. 76, 1, p. 103-106 4 p.Research output: Contribution to journal › Article › peer-review
40 Scopus citations -
New cytotoxic 1,2,4-thiadiazole alkaloids from the ascidian Polycarpa aurata
Pham, C. D., Weber, H., Hartmann, R., Wray, V., Lin, W., Lai, D. & Proksch, P., May 3 2013, In: Organic Letters. 15, 9, p. 2230-2233 4 p.Research output: Contribution to journal › Article › peer-review
47 Scopus citations